Publications


Long-Term Exposure to Sucrose during the Differentiation Process Increases Permeability Independently of TAS1R3 in In Vitro Models of the Intestinal Barrier Function
Journal of Agricultural and Food Chemistry
2025-07-30 | Journal article
DOI: 10.1021/acs.jafc.5c02797
Contributors: Markus L. Rechl; Evelin Balika; Sascha Oberle; Verena Preinfalk; Sarah Stadlmayr; Jana Rasztovits; Jakob P. Ley; Barbara Lieder

Novel Perspective on the Plasticity of Taste Perception: Is Food- and Exercise-Induced Inflammation Associated with Sweet Taste Sensitivity and Preference?
Journal of Agricultural and Food Chemistry
2024-07-10 | Journal article
DOI: 10.1021/acs.jafc.3c09028
Contributors: Isabella Kimmeswenger; Barbara Lieder

Dipeptidyl-peptidase 4 (DPP4) mediates fatty acid uptake inhibition by glucose via TAS1R3 and GLUT-2 in Caco-2 enterocytes
Heliyon
2024-05 | Journal article
DOI: 10.1016/j.heliyon.2024.e30329
Contributors: Verena Preinfalk; Isabella Kimmeswenger; Veronika Somoza; Barbara Lieder
Development and In Vivo Evaluation of Small-Molecule Ligands for Positron Emission Tomography of Immune Checkpoint Modulation Targeting Programmed Cell Death 1 Ligand 1
Journal of Medicinal Chemistry
2024-03-14 | Journal article
DOI: 10.1021/acs.jmedchem.3c02342
Contributors: Karsten Bamminger; Verena Pichler; Chrysoula Vraka; Tanja Limberger; Boryana Moneva; Katharina Pallitsch; Barbara Lieder; Anna Sophia Zacher; Stefanie Ponti; Katarína Benčurová et al.
On the Road towards Small-Molecule Programmed Cell Death 1 Ligand 1 Positron Emission Tomography Tracers: A Ligand-Based Drug Design Approach
Pharmaceuticals
2023-07-24 | Journal article
DOI: 10.3390/ph16071051
Contributors: Karsten Bamminger; Verena Pichler; Chrysoula Vraka; Tina Nehring; Katharina Pallitsch; Barbara Lieder; Marcus Hacker; Wolfgang Wadsak

Human Gingival Fibroblasts as a Novel Cell Model Describing the Association between Bitter Taste Thresholds and Interleukin-6 Release
Journal of Agricultural and Food Chemistry
2023-04-05 | Journal article
DOI: 10.1021/acs.jafc.2c06979
Contributors: Johanna Tiroch; Andreas Dunkel; Sonja Sterneder; Sofie Zehentner; Maik Behrens; Antonella Di Pizio; Jakob P. Ley; Barbara Lieder; Veronika Somoza

Impact of lactisole on the time-intensity profile of selected sweeteners in dependence of the binding site
Food chemistry: X
2022 | Journal article
DOI: 10.1016/j.fochx.2022.100446
Part of ISSN: 2590-1575
Individual Sweet Taste Perception Influences Salivary Characteristics After Orosensory Stimulation With Sucrose and Noncaloric Sweeteners
Frontiers in nutrition
2022 | Journal article
DOI: 10.3389/fnut.2022.831726
Part of ISSN: 2296-861X
Long-Term Consumption of a Sugar-Sweetened Soft Drink in Combination with a Western-Type Diet Is Associated with Morphological and Molecular Changes of Taste Markers Independent of Body Weight Development in Mice
Nutrients
2022-01-29 | Journal article
DOI: 10.3390/nu14030594
Contributors: Barbara Lieder; Jozef Čonka; Agnes T. Reiner; Victoria Zabel; Dominik Ameur; Mark M. Somoza; Katarína Šebeková; Peter Celec; Veronika Somoza
Bitter Sensing TAS2R50 Mediates the trans-Resveratrol-Induced Anti-inflammatory Effect on Interleukin 6 Release in HGF-1 Cells in Culture
Journal of Agricultural and Food Chemistry
2021-11-17 | Journal article
DOI: 10.1021/acs.jafc.0c07058
Contributors: Johanna Tiroch; Sonja Sterneder; Antonella Di Pizio; Barbara Lieder; Kathrin Hoelz; Ann-Katrin Holik; Marc Pignitter; Maik Behrens; Mark Somoza; Jakob P. Ley et al.
Gastric Serotonin Biosynthesis and Its Functional Role in L-Arginine-Induced Gastric Proton Secretion
International Journal of Molecular Sciences
2021-05-30 | Journal article
DOI: 10.3390/ijms22115881
Contributors: Ann-Katrin Holik; Kerstin Schweiger; Verena Stoeger; Barbara Lieder; Angelika Reiner; Muhammet Zopun; Julia K. Hoi; Nicole Kretschy; Mark M. Somoza; Stephan Kriwanek et al.
Sweetness Perception is not Involved in the Regulation of Blood Glucose after Oral Application of Sucrose and Glucose Solutions in Healthy Male Subjects
Molecular Nutrition & Food Research
2021-01 | Journal article
DOI: 10.1002/mnfr.202000472
Contributors: Verena Grüneis; Kerstin Schweiger; Claudia Galassi; Corinna M. Karl; Julia Treml; Jakob P. Ley; Jürgen König; Gerhard E. Krammer; Veronika Somoza; Barbara Lieder
TRPA1 Agonist Cinnamaldehyde Decreases Adipogenesis in 3T3-L1 Cells More Potently than the Non-agonist Structural Analog Cinnamyl Isobutyrate
ACS Omega
2020-12-29 | Journal article
DOI: 10.1021/acsomega.0c05083
Contributors: Julia K. Hoi; Barbara Lieder; Beatrix Liebisch; Christiane Czech; Joachim Hans; Jakob P. Ley; Veronika Somoza
Sweet Taste Antagonist Lactisole Administered in Combination with Sucrose, But Not Glucose, Increases Energy Intake and Decreases Peripheral Serotonin in Male Subjects
Nutrients
2020-10-14 | Journal article
DOI: 10.3390/nu12103133
Contributors: Kerstin Schweiger; Verena Grüneis; Julia Treml; Claudia Galassi; Corinna M. Karl; Jakob P. Ley; Gerhard E. Krammer; Barbara Lieder; Veronika Somoza
Structure-dependent effects of sweet and sweet taste affecting compounds on their sensorial properties
Food Chemistry: X
2020-09 | Journal article
DOI: 10.1016/j.fochx.2020.100100
Contributors: Corinna M. Karl; Martin Wendelin; Dariah Lutsch; Gerhard Schleining; Klaus Dürrschmid; Jakob P. Ley; Gerhard E. Krammer; Barbara Lieder
In Vitro Digestion of Grape Seed Oil Inhibits Phospholipid-Regulating Effects of Oxidized Lipids
Biomolecules
2020-05-02 | Journal article
DOI: 10.3390/biom10050708
Contributors: Sarah Fruehwirth; Sofie Zehentner; Mohammed Salim; Sonja Sterneder; Johanna Tiroch; Barbara Lieder; Martin Zehl; Veronika Somoza; Marc Pignitter
Correction to Structure-Dependent Effects of Cinnamaldehyde Derivatives on TRPA1-Induced Serotonin Release in Human Intestinal Cell Models
Journal of Agricultural and Food Chemistry
2020-04-29 | Journal article
DOI: 10.1021/acs.jafc.0c02180
Contributors: Barbara Lieder; Julia Hoi; Nathalie Burian; Joachim Hans; Ann-Katrin Holik; Leopoldo Raul Beltran Marquez; Jakob P. Ley; Hanns Hatt; Veronika Somoza
Structure-dependent effects of cinnamaldehyde-derivatives on TRPA1 induced serotonin release in human intestinal cell models
Journal of Agricultural and Food Chemistry
2020-03-12 | Journal article
DOI: 10.1021/acs.jafc.9b08163
Part of ISSN: 0021-8561
Part of ISSN: 1520-5118
Identification of Cinnamaldehyde as Most Effective Fatty Acid Uptake Reducing Cinnamon-Derived Compound in Differentiated Caco-2 Cells Compared to Its Structural Analogues Cinnamyl Alcohol, Cinnamic Acid, and Cinnamyl Isobutyrate
Journal of Agricultural and Food Chemistry
2019 | Journal article
DOI: 10.1021/acs.jafc.9b04274
EID: 2-s2.0-85073763898
Contributors: Hoi, J.K.; Lieder, B.; Pignitter, M.; Hans, J.; Ley, J.P.; Lietard, J.; Hoelz, K.; Somoza, M.; Somoza, V.
Wheat Protein Hydrolysate Fortified With l‐Arginine Enhances Satiation Induced by the Capsaicinoid Nonivamide in Moderately Overweight Male Subjects
Molecular Nutrition & Food Research
2019-12 | Journal article
DOI: 10.1002/mnfr.201900133
Contributors: Verena Stoeger; Barbara Lieder; Johanna Riedel; Kerstin Schweiger; Julia Hoi; Veronika Ruzsanyi; Martin Klieber; Petra Rust; Joachim Hans; Jakob P Ley et al.
Biological Evaluation of Natural and Synthesized Homovanillic Acid Esters as Inhibitors of Intestinal Fatty Acid Uptake in Differentiated Caco-2 Cells
Molecules
2019-10-07 | Journal article
DOI: 10.3390/molecules24193599
Contributors: Barbara Lieder; Joachim Hans; Fabia Hentschel; Katrin Geissler; Jakob Ley
Only aG al bound to lipids, but not to proteins, is transported across enterocytes as an IgE reactive molecule that can induce effector cell activation
Allergy
2019-05-18 | Journal article
DOI: 10.1111/all.13873
Part of ISSN: 0105-4538
Part of ISSN: 1398-9995
Cinnamyl Isobutyrate Decreases Plasma Glucose Levels and Total Energy Intake from a Standardized Breakfast: A Randomized, Crossover Intervention
Molecular Nutrition and Food Research
2018 | Journal article
DOI:   10.1002/mnfr.201701038 
EID: 2-s2.0-85052755728
Contributors: Hochkogler, C.M.; Hoi, J.K.; Lieder, B.; Müller, N.; Hans, J.; Widder, S.; Ley, J.P.; Somoza, V.
Identification of bitter-taste intensity and molecular weight as amino acid determinants for the stimulating mechanisms of gastric acid secretion in human parietal cells in culture.
Journal of agricultural and food chemistry
2018-06 | Journal article
DOI: 10.1021/acs.jafc.8b01802
PMID: 29879844
Contributors: Stoeger V; Liszt KI; Lieder B; Wendelin M; Zopun M; Hans J; Ley JP; Krammer GE; Somoza V
Non-caloric sweeteners induce peripheral serotonin secretion via a T1R3-dependent pathway in human gastric cells in culture.
Journal of agricultural and food chemistry
2018-06 | Journal article
DOI: 10.1021/acs.jafc.8b02071
PMID: 29874909
Contributors: Zopun M; Lieder B; Holik AK; Ley JP; Hans J; Somoza V
Capsaicin and nonivamide similarly modulate outcome measures of mitochondrial energy metabolism in HepG2 and 3T3-L1 cells.
Food & function
2018-02 | Journal article
DOI: 10.1039/c7fo01626c
PMID: 29362767
Contributors: Hochkogler CM; Lieder B; Schachner D; Heiss E; Schröter A; Hans J; Ley JP; Krammer GE; Somoza V
The flavanone homoeriodictyol increases SGLT-1-mediated glucose uptake but decreases serotonin release in differentiated Caco-2 cells.
2017 | Journal article
DOI: 10.1371/journal.pone.0171580
PMID: 28192456
PMC: PMC5305062
Contributors: Lieder B; Hoi JK; Holik AK; Geissler K; Hans J; Friedl B; Liszt K; Krammer GE; Ley JP; Somoza V
The Advanced Glycation End Product N(ϵ) -Carboxymethyllysine and its Precursor Glyoxal Increase Serotonin Release from Caco-2 cells.
Journal of cellular biochemistry
2017-10 | Journal article
DOI: 10.1002/jcb.26439
PMID: 29052845
Appetite-Inducing Effects of Homoeriodictyol: Two Randomized, Cross-Over Interventions.
Molecular nutrition & food research
2017-08 | Journal article
DOI: 10.1002/mnfr.201700459
PMID:   28834253
Caffeine induces gastric acid secretion via bitter taste signaling in gastric parietal cells.
Proceedings of the National Academy of Sciences of the United States of America
2017-07 | Journal article
DOI: 10.1073/pnas.1703728114
PMID: 28696284
PMC: PMC5544304
A 12-week intervention with nonivamide, a TRPV1 agonist, prevents a dietary-induced body fat gain and increases peripheral serotonin in moderately overweight subjects.
2017-05 | Journal article
DOI: 10.1002/mnfr.201600731
PMID: 28012242
Contributors: Hochkogler CM; Lieder B; Rust P; Berry D; Meier SM; Pignitter M; Riva A; Leitinger A; Bruk A; Wagner S et al.
The Alkamide trans-Pellitorine Targets PPARγ via TRPV1 and TRPA1 to Reduce Lipid Accumulation in Developing 3T3-L1 Adipocytes
Frontiers in Pharmacology
2017-05-31 | Journal article
DOI: 10.3389/fphar.2017.00316
Part of ISSN: 1663-9812
Sensory active piperine analogues from Macropiper excelsum and their effects on intestinal nutrient uptake in Caco-2 cells.
2017-03 | Journal article
DOI: 10.1016/j.phytochem.2016.12.016
PMID: 28065397
Contributors: Obst K; Lieder B; Reichelt KV; Backes M; Paetz S; Geißler K; Krammer G; Somoza V; Ley JP; Engel KH
Nonivamide, a capsaicin analogue, exhibits anti-inflammatory properties in peripheral blood mononuclear cells and U-937 macrophages.
2017-02 | Journal article
DOI: 10.1002/mnfr.201600474
PMID: 27666931
Contributors: Walker J; Ley JP; Schwerzler J; Lieder B; Beltran L; Ziemba PM; Hatt H; Hans J; Widder S; Krammer GE et al.
N(ϵ) -Carboxymethyllysine Increases the Expression of miR-103/143 and Enhances Lipid Accumulation in 3T3-L1 Cells.
2016-10 | Journal article
DOI: 10.1002/jcb.25576
PMID: 27137869
PMC: PMC4982050
Contributors: Holik AK; Lieder B; Kretschy N; Somoza MM; Held S; Somoza V
Nonivamide enhances miRNA let-7d expression and decreases adipogenesis PPARγ expression in 3T3-L1 cells.
2015-06 | Journal article
DOI: 10.1002/jcb.25052
PMID: 25704235
PMC: PMC4949678
Contributors: Rohm B; Holik AK; Kretschy N; Somoza MM; Ley JP; Widder S; Krammer GE; Marko D; Somoza V
Capsaicin, nonivamide and trans-pellitorine decrease free fatty acid uptake without TRPV1 activation and increase acetyl-coenzyme A synthetase activity in Caco-2 cells.
2015-01 | Journal article
DOI: 10.1039/c4fo00435c
PMID: 25422952
Contributors: Rohm B; Riedel A; Ley JP; Widder S; Krammer GE; Somoza V
Structure-dependent effects of pyridine derivatives on mechanisms of intestinal fatty acid uptake: regulation of nicotinic acid receptor and fatty acid transporter expression.
2014-07 | Journal article
DOI: 10.1016/j.jnutbio.2014.03.002
PMID: 24767308
Contributors: Riedel A; Lang R; Rohm B; Rubach M; Hofmann T; Somoza V
The capsaicin analog nonivamide decreases total energy intake from a standardized breakfast and enhances plasma serotonin levels in moderately overweight men after administered in an oral glucose tolerance test: a randomized, crossover trial.
2014-06 | Journal article
DOI: 10.1002/mnfr.201300821
PMID: 24753478
Contributors: Hochkogler CM; Rohm B; Hojdar K; Pignitter M; Widder S; Ley JP; Krammer GE; Somoza V
Nonivamide, a capsaicin analog, increases dopamine and serotonin release in SH-SY5Y cells via a TRPV1-independent pathway.
2013-11 | Journal article
DOI: 10.1002/mnfr.201200846
PMID: 23929722
Contributors: Rohm B; Holik AK; Somoza MM; Pignitter M; Zaunschirm M; Ley JP; Krammer GE; Somoza V
Simultaneous light-directed synthesis of mirror-image microarrays in a photochemical reaction cell with flare suppression.
2013-09 | Journal article
DOI: 10.1021/ac4024318
PMID: 23968455
PMC: PMC3776564
Contributors: Sack M; Kretschy N; Rohm B; Somoza V; Somoza MM
N(ε)-Carboxymethyllysine (CML), a Maillard reaction product, stimulates serotonin release and activates the receptor for advanced glycation end products (RAGE) in SH-SY5Y cells.
2013-07 | Journal article
DOI: 10.1039/c3fo60097a
PMID: 23759926
Contributors: Holik AK; Rohm B; Somoza MM; Somoza V
Biosynthesis of the respiratory toxin bongkrekic acid in the pathogenic bacterium Burkholderia gladioli.
2012-09 | Journal article
DOI: 10.1016/j.chembiol.2012.07.022
PMID: 22999884
Contributors: Moebius N; Ross C; Scherlach K; Rohm B; Roth M; Hertweck C
Caffeine dose-dependently induces thermogenesis but restores ATP in HepG2 cells in culture.
2012-09 | Journal article
DOI: 10.1039/c2fo30053b
PMID: 22710994
Contributors: Riedel A; Pignitter M; Hochkogler CM; Rohm B; Walker J; Bytof G; Lantz I; Somoza V
Identification of coffee components that stimulate dopamine release from pheochromocytoma cells (PC-12)
Food and Chemical Toxicology
2012-02 | Journal article
DOI: 10.1016/j.fct.2011.09.041
Part of ISSN: 0278-6915
Biosynthesis of the mitochondrial adenine nucleotide translocase (ATPase) inhibitor bongkrekic acid in Burkholderia gladioli.
2010-04 | Journal article
DOI: 10.1039/b925483h
PMID: 20237660
Contributors: Rohm B; Scherlach K; Hertweck C
Toxin production by bacterial endosymbionts of a Rhizopus microsporus strain used for tempe/sufu processing.
2010-01 | Journal article
DOI: 10.1016/j.ijfoodmicro.2009.10.010
PMID: 19942312
Contributors: Rohm B; Scherlach K; Möbius N; Partida-Martinez LP; Hertweck C